Development of inhibitors for the enzyme IspF using high-throughput screening and structure-based design
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Author
Date
2011Type
- Doctoral Thesis
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https://doi.org/10.3929/ethz-a-006831277Publication status
publishedExternal links
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Contributors
Examiner: Diederich, François
Examiner: Borschberg, Hans-Jürg
Examiner: Bacher, Adelbert
Publisher
ETH ZurichSubject
ARZNEIMITTELENTWICKLUNG + ARZNEIMITTELDESIGN + ARZNEIMITTELENTDECKUNG; ANTIMALARIA-MITTEL (PHARMAZIE); ENZYMINHIBITOREN (BIOCHEMIE); KOMBINATORISCHE CHEMIE + KOMBINATORISCHE SYNTHESE; STRUKTUR-WIRKUNG BEZIEHUNG, CHEMISCHE EINFLÜSSE AUF ARZNEIMITTELWIRKUNG (PHARMAKOLOGIE); PYRIMIDIN UND DERIVATE (HETEROCYCLISCHE KOHLENWASSERSTOFFE); SULFONAMIDE (PHARMAZIE); DRUG DEVELOPMENT + DRUG DESIGN + DRUG DISCOVERY (PHARMACY); ANTIMALARIALS (PHARMACY); ENZYME INHIBITORS (BIOCHEMISTRY); COMBINATORIAL CHEMISTRY + COMBINATORIAL SYNTHESIS; STRUCTURE-ACTIVITY RELATIONSHIP + CHEMICAL INFLUENCE ON DRUG ACTION (PHARMACOLOGY); PYRIMIDINE AND DERIVATIVES (HETEROCYCLIC HYDROCARBONS); SULFONAMIDES (PHARMACY)Organisational unit
03344 - Diederich, François (emeritus)
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